Patent details

EP2637661 Title: Use of (S)-pyrrolidine-1,2-dicarboxylic acid 2-amide 1-({4-methyl-5-[2-(2,2,2-trifluoro-1,1-dimethyl-ethyl)- pyridin-4-yl]-thiazol-2-yl}-amide) in the treatment of EGFR dependent diseases or diseases that have acquired resistance to agents that target EGFR family members

Basic Information

Publication number:
EP2637661
PCT Application Number:
EP2011069522
Type:
European Patent Granted for LU
Legal Status:
Lapsed
Application number:
EP117821116
PCT Publication Number:
WO2012062694
First applicant's nationality:
Translation Language:
EPO Publication Language:
English
English Title of Invention:
Use of (S)-pyrrolidine-1,2-dicarboxylic acid 2-amide 1-({4-methyl-5-[2-(2,2,2-trifluoro-1,1-dimethyl-ethyl)- pyridin-4-yl]-thiazol-2-yl}-amide) in the treatment of EGFR dependent diseases or diseases that have acquired resistance to agents that target EGFR family members
French Title of Invention:
Utilisation de la 1-({4-méthyl-5-[2-(2,2,2-trifluoro- 1,1-diméthyléthyl)- pyridin-4-yl]thiazole-2-yl}-amide) du 2-amide de l'acide (S)-pyrrolidine-1,2-dicarboxylique dans le traitement de maladies dépendantes d'EGFR ou de maladies qui ont acquis une résistance aux agents qui ciblent des membres de la famille d'EGFR
German Title of Invention:
Verwendung von (S)-Pyrrolidin-1,2-Dicarbonsäure-2-Amid 1 - ({4-Methyl-5- [2- (2,2,2-Trifluor-1,1-Dimethylethyl)Pyridin-4- yl] Thiazol-2-yl}Amid) zur Behandlung von EGFR-abhängigen Erkrankungen oder Erkrankungen mit erworbener Resistenz gegenüber Wirkstoffen, die auf EGFR-Familienmitglieder gerichtet sind
SPC Number:

Dates

Filing date:
07/11/2011
Grant date:
20/12/2017
EP Publication Date:
18/09/2013
PCT Publication Date:
18/05/2012
Claims Translation Received Date:
Translations Received Date (B1 EP Publication):
Translations Received Date (B2 EP Publication):
Translations Received Date (B3 EP Publication):
Publication date:
20/12/2017
EP B1 Publication Date:
20/12/2017
EP B2 Publication Date:
EP B3 Publication Date:
Lapsed date:
07/11/2018
Expiration date:
07/11/2031
Renunciation date:
Revocation date:
Annulment date:

Owner

From:
13/12/2017
 
 

Name:
Novartis AG
Address:
Lichtstrasse 35, 4056 Basel, Switzerland (CH)

Inventor

1

Name:
MAIRA, Sauveur-Michel
Address:
Switzerland (CH)

2

Name:
SCHNELL, Christian René
Address:
Switzerland (CH)

3

Name:
GARCIA-ECHEVERRIA, Carlos
Address:
France (FR)

4

Name:
FRITSCH, Christine
Address:
Switzerland (CH)

5

Name:
BRACHMANN, Saskia Maria
Address:
Switzerland (CH)

Priority

Priority Number:
411117 P
Priority Date:
08/11/2010
Priority Country:
United States (US)

Classification

IPC classification:
A61K 31/4439; A61K 31/517; A61K 39/00; A61K 39/395; A61K 45/06; A61P 35/00; C07K 16/32;

Publication

European Patent Bulletin

Issue number:
201751
Publication date:
20/12/2017
Description:
Grant (B1)

Annual Fees

Annual Fee Due Date:
Annual Fee Number:
Expected Payer:
Last Annual Fee Payment Date:
Last Annual Fee Paid Number:
Payer:
Filing date Document type Number of pages
30/03/2019 Outgoing Correspondence 1