Patent details

EP3524601 Title: N-{3-[3-CYCLOPROPYL-5-(2-FLUORO-4-IODOPHENYLAMINO)-6,8-DIMETHYL-2,4,7-TRIOXO-3,4,6,7-TETRAHYDRO-2H-PYRIDO[4,3-D]PYRIMIDIN-1-YL]-PHENYL}-CYCLOPROPANECARBOXAMIDE DIMETHYL SULPHOXIDE SOLVATE AS AN MEK1/2 INHIBITOR

Basic Information

Publication number:
EP3524601
PCT Application Number:
RU2016000862
Type:
European Patent Granted for LU
Legal Status:
Lapsed
Application number:
EP169187630
PCT Publication Number:
WO2018070900
First applicant's nationality:
Translation Language:
EPO Publication Language:
English
English Title of Invention:
N-{3-[3-CYCLOPROPYL-5-(2-FLUORO-4-IODOPHENYLAMINO)-6,8-DIMETHYL-2,4,7-TRIOXO-3,4,6,7-TETRAHYDRO-2H-PYRIDO[4,3-D]PYRIMIDIN-1-YL]-PHENYL}-CYCLOPROPANECARBOXAMIDE DIMETHYL SULPHOXIDE SOLVATE AS AN MEK1/2 INHIBITOR
French Title of Invention:
SOLVATE DE DIMÉTHYLSULFOXYDE N-{3-[3-CYCLOPROPYL-5-(2-FLUORO-4-IODOPHÉNYLAMINO)-6,8-DIMÉTHYL-2,4,7-TRIOXO-3,4,6,7-TÉTRAHYDRO-2N-PYRIDO[4,3-D]PYRIMIDIN-1-YL]-PHÉNYL}- CYCLOPROPANECARBOXAMIDE UTILISÉ EN TANT QUE INHIBITEUR DE MEK1/2
German Title of Invention:
N-{3-[3-CYCLOPROPYL-5-(2-FLUOR-4-IODOPHENYLAMINO)-6,8-DIMETHYL-2,4,7-TRIOXO-3,4,6,7-TETRAHYDRO-2H-PYRIDO[4,3-D]PYRIMIDIN-1-YL]-PHENYL}-CYCLOPROPANCARBOXAMID-DIMETHYLSULFOXID-SOLVAT ALS MEK1/2-INHIBITOR
SPC Number:

Dates

Filing date:
12/12/2016
Grant date:
13/10/2021
EP Publication Date:
14/08/2019
PCT Publication Date:
19/04/2018
Claims Translation Received Date:
Translations Received Date (B1 EP Publication):
Translations Received Date (B2 EP Publication):
Translations Received Date (B3 EP Publication):
Publication date:
13/10/2021
EP B1 Publication Date:
13/10/2021
EP B2 Publication Date:
EP B3 Publication Date:
Lapsed date:
12/12/2022
Expiration date:
12/12/2036
Renunciation date:
Revocation date:
Annulment date:

Owner

From:
06/10/2021
 
 

Name:
R-Pharm Joint Stock Company (R-Pharm, JSC)
Address:
Berzarina str. 19 bld. 1, Moscow 123154, Russian Federation (RU)

Name:
Repik, Alexey Evgenievich
Address:
54 Kotoroslnaya nab., Apt. 9, Yaroslavl, 150000, Russian Federation (RU)

Agent

Name:
VALIPAT
From:
25/10/2021
Address:
Uitbreidingstraat 72-5, 2600, Antwerp, Belgium (BE)
To:

Inventor

1

Name:
CHAFEEV, Mikhail Airatovich
Address:
Russian Federation (RU)

2

Name:
IVACHTCHENKO, Alexandre Vasilievich
Address:
United States (US)

3

Name:
IGNATIEV, Vasily Gennadievich
Address:
Russian Federation (RU)

4

Name:
REPIK, Alexey Evgenievich
Address:
Russian Federation (RU)

Priority

Priority Number:
2016139641
Priority Date:
10/10/2016
Priority Country:
Russian Federation (RU)

Classification

IPC classification:
C07D 471/04; A61P 35/00; A61K 31/519;

Publication

European Patent Bulletin

Issue number:
202141
Publication date:
13/10/2021
Description:
Grant (B1)

Deed

Power of attorney

Change Kind/ Decision Type:
Assignment
Deed Number:
RC20210000455A
Date Registered:
25/10/2021
Licence Effective Date:
Licence Expiration Date:
Scope of Licence:
Deed Filer:
VALIPAT
Journal Edition Number:
Text:
Constitution de mandataire
Country Code:
Updated Licence Number:
Terminated Licence Number:

Removed Pledgee

Name:
Address:

Annual Fees

Annual Fee Due Date:
Annual Fee Number:
Expected Payer:
Last Annual Fee Payment Date:
30/11/2021
Last Annual Fee Paid Number:
6
Last Annual Fee Paid Amount:
66 Euro
Payer:
Renewalsdesk Limited
Filing date Document type Number of pages
25/10/2021 Request For Change 2
25/10/2021 Outgoing Correspondence 2