Patent details

EP3089961 Title: PROCESS FOR THE MANUFACTURE OF (E)-4-N,N-DIALKYLAMINO CROTONIC ACID IN HX SALT FORM AND USE THEREOF FOR SYNTHESIS OF EGFR TYROSINE KINASE INHIBITORS

Basic Information

Publication number:
EP3089961
PCT Application Number:
EP2014079150
Type:
European Patent Granted for LU
Legal Status:
Lapsed
Application number:
EP148280373
PCT Publication Number:
WO2015101554
First applicant's nationality:
Translation Language:
EPO Publication Language:
English
English Title of Invention:
PROCESS FOR THE MANUFACTURE OF (E)-4-N,N-DIALKYLAMINO CROTONIC ACID IN HX SALT FORM AND USE THEREOF FOR SYNTHESIS OF EGFR TYROSINE KINASE INHIBITORS
French Title of Invention:
PROCÉDÉ DE FABRICATION D'ACIDE (E)-4-N,N-DIALKYLAMINOCROTONIQUE SOUS FORME DE SEL HX ET SON UTILISATION POUR LA SYNTHÈSE D'INHIBITEURS D'EGFR TYROSINE KINASE
German Title of Invention:
VERFAHREN ZUR HERSTELLUNG VON (E)-4-N,N-DIALKYLAMINO-CROTONSÄURE IN HX-SALZFORM UND VERWENDUNG DAVON ZUR SYNTHESE VON EGFR-TYROSINKINASEHEMMERN
SPC Number:

Dates

Filing date:
23/12/2014
Grant date:
11/07/2018
EP Publication Date:
09/11/2016
PCT Publication Date:
09/07/2015
Claims Translation Received Date:
Translations Received Date (B1 EP Publication):
Translations Received Date (B2 EP Publication):
Translations Received Date (B3 EP Publication):
Publication date:
11/07/2018
EP B1 Publication Date:
11/07/2018
EP B2 Publication Date:
EP B3 Publication Date:
Lapsed date:
23/12/2018
Expiration date:
23/12/2034
Renunciation date:
Revocation date:
Annulment date:

Owner

From:
04/07/2018
 
 

Name:
Boehringer Ingelheim International GmbH
Address:
Binger Strasse 173, 55216 Ingelheim am Rhein, Germany (DE)

Inventor

1

Name:
DENG, Da
Address:
China (CN)

2

Name:
ZHENG, Juncheng
Address:
China (CN)

3

Name:
LV, Guanghua
Address:
China (CN)

4

Name:
KROEBER, Jutta
Address:
Germany (DE)

5

Name:
BRANDENBURG, Joerg
Address:
Germany (DE)

6

Name:
YAN, Jun
Address:
China (CN)

7

Name:
SCHOLZ, Ulrich
Address:
Germany (DE)

Priority

Priority Number:
PCT/CN2013/091071
Priority Date:
31/12/2013
Priority Country:
World Intellectual Property Office (WIPO) (WO)

Classification

IPC classification:
C07C 227/10; C07C 227/18; C07C 229/30; C07D 405/04;

Publication

European Patent Bulletin

Issue number:
201828
Publication date:
11/07/2018
Description:
Grant (B1)

Annual Fees

Annual Fee Due Date:
Annual Fee Number:
Expected Payer:
Last Annual Fee Payment Date:
Last Annual Fee Paid Number:
Payer:
Filing date Document type Number of pages
30/04/2019 Outgoing Correspondence 1